Suppositories with a lot of phytocannabinoid acids

Peter Vermeul: Lately we have been inundated with questions from people with prostate problems, among other things, whether suppositories can be a solution? According to the specialists I regularly speak to, this could well have something to do with the aftermath of the Covid pandemic, but that is besides the point.   

In a short period of time, I have helped several people, at their request – with the knowledge and in consultation with the treating physicians – to make their own suppositories with a high percentage of phytocannabinoid acids such as CBDa, CBGa, etc.

The big advantage of these full-spectrum extracts is that it is much better absorbed into the bloodstream than the decarboxylated (heated) form.

No psychoactive effect with these suppositories

A large number of people quickly let me know that it went very positively and that the doctors were amazed. But one swallow does not make a summer and time will tell how it will turn out.

Cannabis suppositories, whether anal or vaginal, may seem like a strange concept to most, but the benefits far outweigh the drawbacks, making it a fantastic way to experience the tremendous health benefits of cannabis.

Cannabis suppositories are also a dream for medical cannabis patients looking for ways to avoid the psychoactive effects of marijuana (i.e. THC).

The Benefits of Cannabis Suppositories

For decades, suppositories have been used to administer various medications to patients. The pelvic region is home to hundreds of nerves that spread into the legs and spine, while the large intestine also contains ECS receptors . 

Anal cannabis suppositories can be used to treat hemorrhoids, inflammation, Crohn's disease, anal fissures , prostate disorders, restless leg syndrome, sciatica, digestive disorders , and postoperative pain .

Vaginal suppositories can be used by women to help with abdominal pain, cramps, endometriosis , vaginal dryness, inflammation, pre- and post-coital pain, and to relieve menstrual pain.

But no matter what the problems are, rectal suppositories are usually effective throughout the body, especially for problems such as:

• Epileptic seizures where oral dosing is not possible
• Having trouble swallowing medication
• Medication rather not smoking

Unable to keep fluids or pills down due to vomiting/nausea (such as in people undergoing chemotherapy)

Faster absorption of cannabinoids

When the cannabinoids are absorbed through the rectal mucosa, it helps to quickly distribute them to the bloodstream and nearby organs. And it is also an efficient way to eliminate the “high” caused by THC. 

We should note that decarboxylated cannabinoids are generally poorly absorbed into the bloodstream. Especially when using suppositories, it is desirable to use a pure full-spectrum extract, in which the terpenes, flavonoids and phytocannabinoid acids (the non-decarboxylated form) are present in high concentrations.

The absorbability of THCa, CBDa, CBGa (acid form) in the bloodstream is many times higher than the decarboxylated THC, CBD, CBG. 

How to use cannabis suppositories? 

Cannabis suppositories should be stored in the freezer or refrigerator. The cold temperatures are necessary to keep them firm for insertion. Most suppositories are based on coconut oil and/or cocoa butter, which softens and liquefies very quickly at body temperature. 

So speed during insertion is required, otherwise the suppository will become too soft!

To insert rectally, lie on your side and pull your knees up to your chest. Insert the suppository through the rectum using your index finger. It should be inserted about 4 cm to reach the anal sphincter.

You also need to be careful that it doesn't slip away; you can prevent this by clenching the muscles of your buttocks together for about 5 seconds. Then stay in the lying position for at least another five minutes.

There is a possibility that some fluid will leak out later  leaking from the rectum, so it is ideal to use suppositories before going to bed, or when you can free up time to spend the rest of the day at home and relax. To prevent soiling of the bed, it is wise to take measures such as a sanitary towel or old towel.

Different kind of high

For anyone who has never tried a suppository before, it may feel a little strange at first. But it is an excellent way to harness the healing benefits of the cannabis plant, especially for patients who need them most but are unable to consume them in other forms. 

The active substances (cannabinoids, terpenes, flavonoids) in cannabis reach the bloodstream without having to pass through the liver and upper gastrointestinal tract. This results in much higher cannabinoid concentrations – up to 75% –  that are absorbed into the body.

The liver is also essential for getting high/stoned , as THC passes through the liver before reaching the brain to give you the “high.” The best way to describe this absorption, which you might get from suppositories that do contain THC, is one that gives you more of a clear-headed, relaxed feeling.

Peter Vermeul

Owner, Grower, Producer CBD Spain

If you have any questions following this article, please do not hesitate to contact CBD & Herb!